CausalSentinel

Protein Dossier — HMGCR (3-hydroxy-3-methylglutaryl-coenzyme A reductase)

MR feasibility tier: B — No published MR estimate in this resource, BUT a pQTL GWAS exists - instruments are derivable, so a two-sample MR could be run. The upstream is waiting.

1. Published MR estimates (retrieved, not computed)

None in the EpiGraphDB pQTL resource. Absence of an estimate is not evidence of no effect.

2. pQTL instrument availability (Tier-B probe)

Dataset Trait Author Year
prot-c-5230_99_3 HMGR Suhre K 2019

Instruments exist but no MR estimate is in this resource — a two-sample MR here is un-run work.

3. GWAS Catalog results — traits with signal at this locus

855 association rows across 463 traits (831 genome-wide significant rows). Associations are loci, not causal claims; the mapped gene at a locus is not necessarily the effector gene.

Trait best p lead SNP n assoc study MR status
Low density lipoprotein cholesterol levels 1e-602 rs12916 46 GCST90239655 no MR -> candidate analysis
Total cholesterol levels 2e-546 rs12916 51 GCST90239673 no MR -> candidate analysis
Low-density lipoprotein levels 8e-401 rs10942734 1 GCST90662892 no MR -> candidate analysis
Non-HDL cholesterol levels 2e-399 rs12916 5 GCST90239667 no MR -> candidate analysis
LDL cholesterol levels 2e-187 rs12916 13 GCST010245 no MR -> candidate analysis
Direct low density lipoprotein levels (UKB data field 30780) 5e-176 rs12916 1 GCST90468080 no MR -> candidate analysis
LDL cholesterol 5e-173 rs12916 11 GCST90018961 no MR -> candidate analysis
Cholesterol levels (UKB data field 30690) 9e-165 rs12916 1 GCST90468066 no MR -> candidate analysis
low density lipoprotein cholesterol (LDLC, maximum, inv-norm 2e-164 rs12916 3 GCST90475412 no MR -> candidate analysis
low density lipoprotein cholesterol (LDLC, mean, inv-norm tr 2e-160 rs12916 3 GCST90475416 no MR -> candidate analysis
total cholesterol (mean, inv-norm transformed) 8e-155 rs12916 3 GCST90476424 no MR -> candidate analysis
total cholesterol (maximum, inv-norm transformed) 6e-150 rs12916 3 GCST90476420 no MR -> candidate analysis
…and 451 more traits (see JSON)          

4. Phenome map — where this gene is a genetic locus, vs. where MR exists

Top diseases by Open Targets association (of 1080 total). Associations are loci, not causal claims. The causal-status column is a four-state triage per pair: established (curated) = a curated clinical assertion exists (ClinGen/G2P/GEL/Orphanet/ClinVar — any validity level, MR adds little); exploratory rare-variant signal = ExWAS burden evidence without curation — a candidate NEW gene-disease relationship; common-variant locus = GWAS signal, classic pQTL-MR territory; multi-layer = burden+GWAS together, an allelic-series candidate (the strongest causal setup). Burden estimand is carrier-vs-noncarrier, not per-SD MR.

Disease genetic assoc. burden (ExWAS) causal status MR status
Hypercholesterolemia 0.857 common-variant locus no MR -> candidate analysis
hyperlipidemia 0.822 common-variant locus no MR -> candidate analysis
coronary artery disorder 0.687 common-variant locus no MR -> candidate analysis
familial hypercholesterolemia 0.616 common-variant locus no MR -> candidate analysis
stroke disorder 0.481 common-variant locus no MR -> candidate analysis
cardiovascular disorder 0.462 common-variant locus no MR -> candidate analysis
muscular dystrophy, limb-girdle, autosomal recessive 28 0.795 established (curated) no MR -> candidate analysis
type 2 diabetes mellitus 0.44 common-variant locus no MR -> candidate analysis
familial hyperlipidemia 0.674 common-variant locus no MR -> candidate analysis
metabolic disease 0.855 common-variant locus no MR -> candidate analysis
metabolic syndrome 0.69 common-variant locus no MR -> candidate analysis
Disorder of lipid metabolism 0.605 common-variant locus no MR -> candidate analysis
diabetes mellitus 0.516 common-variant locus no MR -> candidate analysis

Of the 13 rows above, 13 have no MR estimate in this resource. Across all retrieved diseases for this gene: 0 exploratory rare-variant signal(s), 0 multi-layer (allelic-series candidate) pair(s). Final triage still belongs to a statistical geneticist.

5. Downstream annotation (druggability & safety preview)

Layer Result
ChEMBL druggability 10 known modulators (3-hydroxy-3-methylglutaryl-coenzyme A reductase)
gnomAD constraint pLI=1, LOEUF=0.433 — LoF-INTOLERANT
GWAS Catalog 92 unique SNPs / 177 rows
ClinVar 112 records; 1 pathogenic in sample of 30
PharmGKB/ClinPGx 10 clinical annotations across 6 drugs

Caveats declared by the tools

Sources

Provenance